Drug Targets
Comprehensive drug target database including GPCRs, ion channels, nuclear receptors, kinases, and enzymes.
Browse the pages below for detailed information.
αβ-Hydrolase 12
αβ-Hydrolase 12 — Enzyme drug target in the 2-Acylglycerol ester turnover family.
αβ-Hydrolase 2
αβ-Hydrolase 2 — Enzyme drug target in the 2-Acylglycerol ester turnover family.
αβ-Hydrolase 6
αβ-Hydrolase 6 — Enzyme drug target in the 2-Acylglycerol ester turnover family.
α1A-adrenoceptor
α1A-adrenoceptor — GPCR drug target in the Adrenoceptors family.
α1B-adrenoceptor
α1B-adrenoceptor — GPCR drug target in the Adrenoceptors family.
α1D-adrenoceptor
α1D-adrenoceptor — GPCR drug target in the Adrenoceptors family.
α2A-adrenoceptor
α2A-adrenoceptor — GPCR drug target in the Adrenoceptors family.
α2B-adrenoceptor
α2B-adrenoceptor — GPCR drug target in the Adrenoceptors family.
α2C-adrenoceptor
α2C-adrenoceptor — GPCR drug target in the Adrenoceptors family.
β1-adrenoceptor
β1-adrenoceptor — GPCR drug target in the Adrenoceptors family.
β2-adrenoceptor
β2-adrenoceptor — GPCR drug target in the Adrenoceptors family.
β3-adrenoceptor
β3-adrenoceptor — GPCR drug target in the Adrenoceptors family.
δ receptor
δ receptor — GPCR drug target in the Opioid receptors family.
γ-Glutamyl carboxylase
γ-Glutamyl carboxylase — Enzyme drug target in the Carboxylases family.
γ-Glutamyltransferase
γ-Glutamyltransferase — Enzyme drug target in the Leukotriene and lipoxin metabolism family.
κ receptor
κ receptor — GPCR drug target in the Opioid receptors family.
μ receptor
μ receptor — GPCR drug target in the Opioid receptors family.
12R-LOX
12R-LOX — Enzyme drug target in the Lipoxygenases family.
12S-LOX
12S-LOX — Enzyme drug target in the Lipoxygenases family.
15-LOX-1
15-LOX-1 — Enzyme drug target in the Lipoxygenases family.
15-LOX-2
15-LOX-2 — Enzyme drug target in the Lipoxygenases family.
3-ketodihydrosphingosine reductase
3-ketodihydrosphingosine reductase — Enzyme drug target in the 3-ketodihydrosphingosine reductase family.
3-Mercaptopyruvate sulfurtransferase
3-Mercaptopyruvate sulfurtransferase — Enzyme drug target in the Hydrogen sulphide synthesis family.
3-phosphoinositide dependent protein kinase 1
3-phosphoinositide dependent protein kinase 1 — Enzyme drug target in the PDK1 family family.
4-aminobutyrate aminotransferase
4-aminobutyrate aminotransferase — Enzyme drug target in the GABA turnover family.
4-hydroxyphenylpyruvate dioxygenase
4-hydroxyphenylpyruvate dioxygenase — Enzyme drug target in the Oxidoreductases family.
4F2hc
4F2hc — Transporter drug target in the SLC3 family family.
5-HT1A receptor
5-HT1A receptor — GPCR drug target in the 5-Hydroxytryptamine receptors family.
5-HT1B receptor
5-HT1B receptor — GPCR drug target in the 5-Hydroxytryptamine receptors family.
5-HT1D receptor
5-HT1D receptor — GPCR drug target in the 5-Hydroxytryptamine receptors family.
5-ht1e receptor
5-ht1e receptor — GPCR drug target in the 5-Hydroxytryptamine receptors family.
5-HT1F receptor
5-HT1F receptor — GPCR drug target in the 5-Hydroxytryptamine receptors family.
5-HT2A receptor
5-HT2A receptor — GPCR drug target in the 5-Hydroxytryptamine receptors family.
5-HT2B receptor
5-HT2B receptor — GPCR drug target in the 5-Hydroxytryptamine receptors family.
5-HT2C receptor
5-HT2C receptor — GPCR drug target in the 5-Hydroxytryptamine receptors family.
5-HT4 receptor
5-HT4 receptor — GPCR drug target in the 5-Hydroxytryptamine receptors family.
5-HT5A receptor
5-HT5A receptor — GPCR drug target in the 5-Hydroxytryptamine receptors family.
5-ht5b receptor
5-ht5b receptor — GPCR drug target in the 5-Hydroxytryptamine receptors family.
5-HT6 receptor
5-HT6 receptor — GPCR drug target in the 5-Hydroxytryptamine receptors family.
5-HT7 receptor
5-HT7 receptor — GPCR drug target in the 5-Hydroxytryptamine receptors family.
5-LOX
5-LOX — Enzyme drug target in the Lipoxygenases family.
5-methyltetrahydrofolate-homocysteine methyltransferase
5-methyltetrahydrofolate-homocysteine methyltransferase — Enzyme drug target in the Methionine turnover family.
5'-nucleotidase IA
5'-nucleotidase IA — Enzyme drug target in the Adenosine turnover family.
5'-nucleotidase IB
5'-nucleotidase IB — Enzyme drug target in the Adenosine turnover family.
5'-nucleotidase II
5'-nucleotidase II — Enzyme drug target in the Adenosine turnover family.
5'-nucleotidase III
5'-nucleotidase III — Enzyme drug target in the Adenosine turnover family.
5'(3')-nucleotidase
5'(3')-nucleotidase — Enzyme drug target in the Adenosine turnover family.
6-phosphofructo-2-kinase/fructose-2,6-biphosphatase 3
6-phosphofructo-2-kinase/fructose-2,6-biphosphatase 3 — Enzyme drug target in the Sugar phosphatases family.
8-oxoguanine DNA glycosylase
8-oxoguanine DNA glycosylase — Enzyme drug target in the DNA glycosylases family.
A-Raf proto-oncogene, serine/threonine kinase
A-Raf proto-oncogene, serine/threonine kinase — Enzyme drug target in the RAF family family.
A1 receptor
A1 receptor — GPCR drug target in the Adenosine receptors family.
A2A receptor
A2A receptor — GPCR drug target in the Adenosine receptors family.
A2B receptor
A2B receptor — GPCR drug target in the Adenosine receptors family.
A3 receptor
A3 receptor — GPCR drug target in the Adenosine receptors family.
aarF domain containing kinase 1
aarF domain containing kinase 1 — Enzyme drug target in the ABC1-B subfamily family.
aarF domain containing kinase 2
aarF domain containing kinase 2 — Enzyme drug target in the ABC1-A subfamily family.
aarF domain containing kinase 5
aarF domain containing kinase 5 — Enzyme drug target in the ABC1-B subfamily family.
ABCA1
ABCA1 — Transporter drug target in the ABCA subfamily family.
ABCA10
ABCA10 — Transporter drug target in the ABCA subfamily family.
ABCA12
ABCA12 — Transporter drug target in the ABCA subfamily family.