Pharmaceutical Chemistry

Drug Targets

Comprehensive drug target database including GPCRs, ion channels, nuclear receptors, kinases, and enzymes.

Browse the pages below for detailed information.

monoacylglycerol lipase

monoacylglycerol lipase — Enzyme drug target in the S33: Prolyl aminopeptidase family.

monoacylglycerol O-acyltransferase 2

monoacylglycerol O-acyltransferase 2 — Enzyme drug target in the Acyltransferases family.

Monoamine oxidase A

Monoamine oxidase A — Enzyme drug target in the Catecholamine turnover family.

Monoamine oxidase B

Monoamine oxidase B — Enzyme drug target in the Catecholamine turnover family.

Monocarboxylate transporter 1

Monocarboxylate transporter 1 — Transporter drug target in the SLC16 family of monocarboxylate transporters family.

Monocarboxylate transporter 10

Monocarboxylate transporter 10 — Transporter drug target in the SLC16 family of monocarboxylate transporters family.

Monocarboxylate transporter 11

Monocarboxylate transporter 11 — Transporter drug target in the SLC16 family of monocarboxylate transporters family.

Monocarboxylate transporter 12

Monocarboxylate transporter 12 — Transporter drug target in the SLC16 family of monocarboxylate transporters family.

Monocarboxylate transporter 13

Monocarboxylate transporter 13 — Transporter drug target in the SLC16 family of monocarboxylate transporters family.

Monocarboxylate transporter 14

Monocarboxylate transporter 14 — Transporter drug target in the SLC16 family of monocarboxylate transporters family.

Monocarboxylate transporter 2

Monocarboxylate transporter 2 — Transporter drug target in the SLC16 family of monocarboxylate transporters family.

Monocarboxylate transporter 3

Monocarboxylate transporter 3 — Transporter drug target in the SLC16 family of monocarboxylate transporters family.

Monocarboxylate transporter 4

Monocarboxylate transporter 4 — Transporter drug target in the SLC16 family of monocarboxylate transporters family.

Monocarboxylate transporter 5

Monocarboxylate transporter 5 — Transporter drug target in the SLC16 family of monocarboxylate transporters family.

Monocarboxylate transporter 6

Monocarboxylate transporter 6 — Transporter drug target in the SLC16 family of monocarboxylate transporters family.

Monocarboxylate transporter 7

Monocarboxylate transporter 7 — Transporter drug target in the SLC16 family of monocarboxylate transporters family.

Monocarboxylate transporter 8

Monocarboxylate transporter 8 — Transporter drug target in the SLC16 family of monocarboxylate transporters family.

Monocarboxylate transporter 9

Monocarboxylate transporter 9 — Transporter drug target in the SLC16 family of monocarboxylate transporters family.

MOS proto-oncogene, serine/threonine kinase

MOS proto-oncogene, serine/threonine kinase — Enzyme drug target in the MOS family family.

motilin receptor

motilin receptor — GPCR drug target in the Motilin receptor family.

mPGES1

mPGES1 — Enzyme drug target in the Prostaglandin synthases family.

mPGES2

mPGES2 — Enzyme drug target in the Prostaglandin synthases family.

MRGPRD

MRGPRD — GPCR drug target in the Class A Orphans with emerging pharmacology family.

MRGPRE

MRGPRE — GPCR drug target in the Class A Orphans with emerging pharmacology family.

MRGPRF

MRGPRF — GPCR drug target in the Class A Orphans with no pharmacology family.

MRGPRG

MRGPRG — GPCR drug target in the Class A Orphans with no pharmacology family.

MRGPRX1

MRGPRX1 — GPCR drug target in the Class A Orphans with emerging pharmacology family.

MRGPRX2

MRGPRX2 — GPCR drug target in the Class A Orphans with emerging pharmacology family.

MRGPRX3

MRGPRX3 — GPCR drug target in the Class A Orphans with no pharmacology family.

MRGPRX4

MRGPRX4 — GPCR drug target in the Class A Orphans with emerging pharmacology family.

MT1 receptor

MT1 receptor — GPCR drug target in the Melatonin receptors family.

MT2 receptor

MT2 receptor — GPCR drug target in the Melatonin receptors family.

Multidrug and toxin extrusion

Multidrug and toxin extrusion — Transporter drug target in the SLC47 family of multidrug and toxin extrusion transporters family.

myeloperoxidase

myeloperoxidase — Enzyme drug target in the Oxidoreductases family.

myosin heavy chain 9

myosin heavy chain 9 — Enzyme drug target in the Myosin heavy chains, class II (MYH) family.

myosin IIIA

myosin IIIA — Enzyme drug target in the NinaC subfamily family.

myosin IIIB

myosin IIIB — Enzyme drug target in the NinaC subfamily family.

myosin light chain kinase

myosin light chain kinase — Enzyme drug target in the Myosin Light Chain Kinase (MLCK) family family.

myosin light chain kinase 2

myosin light chain kinase 2 — Enzyme drug target in the Myosin Light Chain Kinase (MLCK) family family.

myosin light chain kinase 3

myosin light chain kinase 3 — Enzyme drug target in the Myosin Light Chain Kinase (MLCK) family family.

myosin light chain kinase family member 4

myosin light chain kinase family member 4 — Enzyme drug target in the Myosin Light Chain Kinase (MLCK) family family.

N-Acetylated α-linked acidic dipeptidase 2

N-Acetylated α-linked acidic dipeptidase 2 — Enzyme drug target in the M28: Aminopeptidase Y family.

N-Acetylated α-linked acidic dipeptidase-like 1

N-Acetylated α-linked acidic dipeptidase-like 1 — Enzyme drug target in the M28: Aminopeptidase Y family.

N-acetyltransferase 8 like

N-acetyltransferase 8 like — Enzyme drug target in the Acyltransferases family.

N-Acylethanolamine acid amidase

N-Acylethanolamine acid amidase — Enzyme drug target in the N-Acylethanolamine turnover family.

N-Acylphosphatidylethanolamine-phospholipase D

N-Acylphosphatidylethanolamine-phospholipase D — Enzyme drug target in the N-Acylethanolamine turnover family.

N-acylsphingosine amidohydrolase 1

N-acylsphingosine amidohydrolase 1 — Enzyme drug target in the Acid ceramidase family.

N-acylsphingosine amidohydrolase 2

N-acylsphingosine amidohydrolase 2 — Enzyme drug target in the Neutral ceramidases family.

N-acylsphingosine amidohydrolase 2B

N-acylsphingosine amidohydrolase 2B — Enzyme drug target in the Neutral ceramidases family.

N-myristoyltransferase 1

N-myristoyltransferase 1 — Enzyme drug target in the N-myristoyltransferases family.

N-myristoyltransferase 2

N-myristoyltransferase 2 — Enzyme drug target in the N-myristoyltransferases family.

Na-Cl symporter

Na-Cl symporter — Transporter drug target in the SLC12 family of cation-coupled chloride transporters family.

Na+/citrate cotransporter

Na+/citrate cotransporter — Transporter drug target in the SLC13 family of sodium-dependent sulphate/carboxylate transporters family.

Na+/dicarboxylate cotransporter 1

Na+/dicarboxylate cotransporter 1 — Transporter drug target in the SLC13 family of sodium-dependent sulphate/carboxylate transporters family.

Na+/dicarboxylate cotransporter 3

Na+/dicarboxylate cotransporter 3 — Transporter drug target in the SLC13 family of sodium-dependent sulphate/carboxylate transporters family.

Na+/sulfate cotransporter

Na+/sulfate cotransporter — Transporter drug target in the SLC13 family of sodium-dependent sulphate/carboxylate transporters family.

NaBC1

NaBC1 — Transporter drug target in the Sodium-dependent HCO3- transporters family.

NAD(P) dependent 3-beta-hydroxysteroid dehydrogenase NSDHL

NAD(P) dependent 3-beta-hydroxysteroid dehydrogenase NSDHL — Enzyme drug target in the Cholesterol biosynthesis pathway family.

NADPH oxidase 1

NADPH oxidase 1 — Enzyme drug target in the NADPH oxidases family.

NADPH oxidase 3

NADPH oxidase 3 — Enzyme drug target in the NADPH oxidases family.