Pharmaceutical Chemistry

Drug Targets

Comprehensive drug target database including GPCRs, ion channels, nuclear receptors, kinases, and enzymes.

Browse the pages below for detailed information.

Anion exchange protein 3

Anion exchange protein 3 — Transporter drug target in the Anion exchangers family.

Anion exchange protein 4

Anion exchange protein 4 — Transporter drug target in the Anion exchangers family.

ANKH inorganic pyrophosphate transport regulator

ANKH inorganic pyrophosphate transport regulator — Transporter drug target in the SLC62 Pyrophosphate transporters family.

ankyrin repeat and kinase domain containing 1

ankyrin repeat and kinase domain containing 1 — Enzyme drug target in the Receptor interacting protein kinase (RIPK) family family.

AP2 associated kinase 1

AP2 associated kinase 1 — Enzyme drug target in the NAK family family.

apelin receptor

apelin receptor — GPCR drug target in the Apelin receptor family.

ARF GTPase 6

ARF GTPase 6 — Enzyme drug target in the RAS subfamily family.

Arginase I

Arginase I — Enzyme drug target in the Arginase family.

Arginase II

Arginase II — Enzyme drug target in the Arginase family.

Arginine:glycine amidinotransferase

Arginine:glycine amidinotransferase — Enzyme drug target in the Arginine:glycine amidinotransferase family.

Arginyl aminopeptidase

Arginyl aminopeptidase — Enzyme drug target in the M1: Aminopeptidase N family.

Arginyl aminopeptidase-like 1

Arginyl aminopeptidase-like 1 — Enzyme drug target in the M1: Aminopeptidase N family.

Asc-type amino acid transporter 1

Asc-type amino acid transporter 1 — Transporter drug target in the SLC7 family family.

ASH1 like histone lysine methyltransferase

ASH1 like histone lysine methyltransferase — Enzyme drug target in the Histone methyltransferases (HMTs) family.

asparaginase

asparaginase — Enzyme drug target in the Carboxylic ester hydrolases family.

AT1 receptor

AT1 receptor — GPCR drug target in the Angiotensin receptors family.

AT2 receptor

AT2 receptor — GPCR drug target in the Angiotensin receptors family.

ATB0,+

ATB0,+ — Transporter drug target in the Glycine transporter subfamily family.

ATM serine/threonine kinase

ATM serine/threonine kinase — Enzyme drug target in the Other PIKK family kinases family.

ATP citrate lyase

ATP citrate lyase — Enzyme drug target in the Citrate metabolism family.

ATP-binding cassette, sub-family C (CFTR/MRP), member 8

ATP-binding cassette, sub-family C (CFTR/MRP), member 8 — Transporter drug target in the ABCC subfamily family.

ATP12A

ATP12A — Transporter drug target in the H+/K+-ATPases family.

ATP4A

ATP4A — Transporter drug target in the H+/K+-ATPases family.

ATP4B

ATP4B — Transporter drug target in the H+/K+-ATPases family.

ATP7A

ATP7A — Transporter drug target in the P1B P-type ATPases: Cu+-ATPases family.

ATP7B

ATP7B — Transporter drug target in the P1B P-type ATPases: Cu+-ATPases family.

ATPase 13A1

ATPase 13A1 — Transporter drug target in the P5 P-type ATPases: Mn2+-ATPases family.

ATPase 13A3

ATPase 13A3 — Transporter drug target in the P5 P-type ATPases: Mn2+-ATPases family.

ATPase 13A4

ATPase 13A4 — Transporter drug target in the P5 P-type ATPases: Mn2+-ATPases family.

ATPase 13A5

ATPase 13A5 — Transporter drug target in the P5 P-type ATPases: Mn2+-ATPases family.

ATPase cation transporting 13A2

ATPase cation transporting 13A2 — Transporter drug target in the P5 P-type ATPases: Mn2+-ATPases family.

ATPase family AAA domain containing 2

ATPase family AAA domain containing 2 — Enzyme drug target in the ATPases family.

ATPase family AAA domain containing 2B

ATPase family AAA domain containing 2B — Enzyme drug target in the ATPases family.

ATR checkpoint kinase

ATR checkpoint kinase — Enzyme drug target in the ATR subfamily family.

aurora kinase A

aurora kinase A — Enzyme drug target in the Aurora kinase (Aur) family family.

aurora kinase B

aurora kinase B — Enzyme drug target in the Aurora kinase (Aur) family family.

aurora kinase C

aurora kinase C — Enzyme drug target in the Aurora kinase (Aur) family family.

autophagy related 4B cysteine peptidase

autophagy related 4B cysteine peptidase — Enzyme drug target in the C54: Aut2 peptidase family.

autotaxin

autotaxin — Enzyme drug target in the LPA synthesis family.

B-Raf proto-oncogene, serine/threonine kinase

B-Raf proto-oncogene, serine/threonine kinase — Enzyme drug target in the RAF family family.

b0,+-type amino acid transporter 1

b0,+-type amino acid transporter 1 — Transporter drug target in the SLC7 family family.

B0AT1

B0AT1 — Transporter drug target in the Neutral amino acid transporter subfamily family.

B0AT2

B0AT2 — Transporter drug target in the Neutral amino acid transporter subfamily family.

B0AT3

B0AT3 — Transporter drug target in the Neutral amino acid transporter subfamily family.

B1 receptor

B1 receptor — GPCR drug target in the Bradykinin receptors family.

B2 receptor

B2 receptor — GPCR drug target in the Bradykinin receptors family.

Basic amino acid carrier

Basic amino acid carrier — Transporter drug target in the Mitochondrial amino acid transporter subfamily family.

Basolateral Na-K-Cl symporter

Basolateral Na-K-Cl symporter — Transporter drug target in the SLC12 family of cation-coupled chloride transporters family.

BB1 receptor

BB1 receptor — GPCR drug target in the Bombesin receptors family.

BB2 receptor

BB2 receptor — GPCR drug target in the Bombesin receptors family.

BB3 receptor

BB3 receptor — GPCR drug target in the Mas1, BB3/Brs3, GPR17 family.

BCR activator of RhoGEF and GTPase

BCR activator of RhoGEF and GTPase — Enzyme drug target in the BCR family family.

beta adrenergic receptor kinase 1

beta adrenergic receptor kinase 1 — Enzyme drug target in the Beta-adrenergic receptor kinases (βARKs) family.

beta adrenergic receptor kinase 2

beta adrenergic receptor kinase 2 — Enzyme drug target in the Beta-adrenergic receptor kinases (βARKs) family.

beta-secretase 1

beta-secretase 1 — Enzyme drug target in the A1: Pepsin family.

beta-secretase 2

beta-secretase 2 — Enzyme drug target in the A1: Pepsin family.

BGT1

BGT1 — Transporter drug target in the GABA transporter subfamily family.

BLK proto-oncogene, Src family tyrosine kinase

BLK proto-oncogene, Src family tyrosine kinase — Enzyme drug target in the Src family family.

BLM RecQ like helicase

BLM RecQ like helicase — Enzyme drug target in the RecQ helicases family.

BLT1 receptor

BLT1 receptor — GPCR drug target in the Leukotriene receptors family.